MEPIRAMINE

Mepiramine (pyrilamine) is an H1antihistamine used for allergic reactions. Side effects include drowsiness, dry mouth, and dizziness. Only GMP materials will be supplied, logistics all according to GDP.

SKU: ebfd3a9392f0 Category: Tag:

Product Description


Mechanism of Action

MEPIRAMINE displays a broad and multiaxis biochemical interaction profile characterised by modulation of enzymatic networks, receptormediated signalling, intracellular ion regulation, mitochondrial bioenergetics and transcriptional pathway governance. Its structural features suggest interactions with catalytic and regulatory proteins, leading to changes in phosphorylation cycles, metabolic flux, mitochondrial redox balance, calciumsignalling behaviour and stressresponse activation. Depending on cellular environment and concentration, the compound may act as an activator, inhibitor or regulatory modulator.

Benefits and Advantages

This compound supports a wide range of , including:

  • Receptorligand affinity profiling and bindingsite mapping
  • Enzymecascade modelling and catalyticdomain interaction studies
  • Mitochondrialfunction assays, oxidativestress evaluation and metabolicflux tracking
  • Transcriptomic, proteomic and metabolomic investigation for pathway mapping
  • Apoptosis / autophagy pathway research and cellularstress modelling
  • Highresolution mechanismofaction studies and SAR exploration

Side Effects and Risks

Potential risks include oxidative imbalance, mitochondrial overload, ionchannel dysregulation, receptor crosstalk, cytoskeletal disruption and dosedependent cytotoxicity. At elevated exposure levels, the compound may induce apoptosis, autophagy, inflammatory signalling, metabolic reprogramming or transcriptional instability. Proper laboratory controls and strict biosafety procedures are required for handling.

Only GMP materials will be supplied, logistics all according to GDP.

Datasheet


Molecular Formula

C17H23N3O

Molecular Weight

285.4 g/mol

CAS Number

91-84-9

Storage Condition

Store in a cool, dry place. Keep container tightly closed. Protect from moisture and light.

Solubility

less than 1 mg/mL at 68 °F (NTP, 1992)

Purity

Purity information is available upon request (COA).

Synonym

Mepyramine; pyrilamine; 91-84-9; Pyranisamine; Dorantamin

IUPAC/Chemical Name

N'-[(4-methoxyphenyl)methyl]-N,N-dimethyl-N'-pyridin-2-ylethane-1,2-diamine

InChl Key

YECBIJXISLIIDS-UHFFFAOYSA-N

InChl Code

InChI=1S/C17H23N3O/c1-19(2)12-13-20(17-6-4-5-11-18-17)14-15-7-9-16(21-3)10-8-15/h4-11H,12-14H2,1-3H3

References

https://pubchem.ncbi.nlm.nih.gov/compound/4992;

3D Conformer.

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