About MedicaPharma
MedicaPharma distributes high-quality active pharmaceutical ingredients (APIs) to hospitals, commercial (compounding) pharmacies, research institutes, and universities worldwide.
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Let us handle your sourcing / supply activities. Highly experienced in sourcing specialty raw pharmaceutical ingredients from niche GMP manufacturers around the world.
Why Choose MedicaPharma
Niche API specialist - Pro-active supply partner - High service level - Global network - Logistics according to GDP regulations
Product Description
Mechanism of Action
Clebopride maleate is a dopamine D receptor antagonist with prokinetic and antiemetic activity. It enhances acetylcholine release in enteric neurons, promoting gastric emptying and intestinal motility. It also reduces nausea through chemoreceptor trigger-zone modulation.
Benefits and Advantages
Used in GImotility research, Dantagonist pathway studies, dyspepsia modelling, gastroparesis investigations and neuroenteric signalmodulation assays.
Side Effects and Risks
Risks include extrapyramidal symptoms, hyperprolactinemia, restlessness, diarrhea and hypotension. Handle as a neuroactive GIprokinetic agent.
Only GMP materials will be supplied, logistics all according to GDP.
Datasheet
| Molecular Formula | C21H24ClN3O6 |
|---|---|
| Molecular Weight | 489.9 g/mol |
| CAS Number | 84370-95-6 |
| Storage Condition | Store in a cool, dry place. Keep container tightly closed. Protect from moisture and light. |
| Solubility | Solubility depends on solvent and conditions (e.g., pH). Please contact us for solvent-specific guidance. |
| Purity | Purity information is available upon request (COA). |
| Synonym | Clebopride maleate; 84370-95-6; DTXSID6047787; P42041X5SU; DTXCID6027767 |
| IUPAC/Chemical Name | 4-amino-N-(1-benzylpiperidin-4-yl)-5-chloro-2-methoxybenzamide;(Z)-but-2-enedioic acid |
| InChl Key | BCVIWCRZYPHHMQ-BTJKTKAUSA-N |
| InChl Code | InChI=1S/C20H24ClN3O2.C4H4O4/c1-26-19-12-18(22)17(21)11-16(19)20(25)23-15-7-9-24(10-8-15)13-14-5-3-2-4-6-14;5-3(6)1-2-4(7)8/h2-6,11-12,15H,7-10,13,22H2,1H3,(H,23,25);1-2H,(H,5,6)(H,7,8)/b;2-1- |
| References |
3D Conformer.
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