About MedicaPharma
MedicaPharma distributes high-quality active pharmaceutical ingredients (APIs) to hospitals, commercial (compounding) pharmacies, research institutes, and universities worldwide.
Network of over +400 GMP API producers
Let us handle your sourcing / supply activities. Highly experienced in sourcing specialty raw pharmaceutical ingredients from niche GMP manufacturers around the world.
Why Choose MedicaPharma
Niche API specialist - Pro-active supply partner - High service level - Global network - Logistics according to GDP regulations
Product Description
Mechanism of Action
Clebopride maleate is a dopamine D₂ receptor antagonist with prokinetic and antiemetic activity. It enhances acetylcholine release in enteric neurons, promoting gastric emptying and intestinal motility. It also reduces nausea through chemoreceptor trigger-zone modulation.
Benefits and Advantages
Used in GI‑motility research, D₂‑antagonist pathway studies, dyspepsia modelling, gastroparesis investigations and neuro‑enteric signal‑modulation assays.
Side Effects and Risks
Risks include extrapyramidal symptoms, hyperprolactinemia, restlessness, diarrhea and hypotension. Handle as a neuroactive GI‑prokinetic agent.
Datasheet
| Molecular Formula | C21H24ClN3O6 |
|---|---|
| Molecular Weight | 489.9 g/mol |
| CAS Number | 84370-95-6 |
| Storage Condition | Store in a cool, dry place. Keep container tightly closed. Protect from moisture and light. |
| Solubility | Solubility depends on solvent and conditions (e.g., pH). Please contact us for solvent-specific guidance. |
| Purity | Purity information is available upon request (COA). |
| Synonym | Clebopride maleate; 84370-95-6; DTXSID6047787; P42041X5SU; DTXCID6027767 |
| IUPAC/Chemical Name | 4-amino-N-(1-benzylpiperidin-4-yl)-5-chloro-2-methoxybenzamide;(Z)-but-2-enedioic acid |
| InChl Key | BCVIWCRZYPHHMQ-BTJKTKAUSA-N |
| InChl Code | InChI=1S/C20H24ClN3O2.C4H4O4/c1-26-19-12-18(22)17(21)11-16(19)20(25)23-15-7-9-24(10-8-15)13-14-5-3-2-4-6-14;5-3(6)1-2-4(7)8/h2-6,11-12,15H,7-10,13,22H2,1H3,(H,23,25);1-2H,(H,5,6)(H,7,8)/b;2-1- |
| References |
3D Conformer.
(Click, turn or enlarge)
Download our GMP API Product List.
MedicaPharma is an EU-based supplier of GMP-certified APIs that serves leading healthcare institutions and research organizations.
Click here to download our full API product list.
