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MedicaPharma distributes high-quality active pharmaceutical ingredients (APIs) to hospitals, commercial (compounding) pharmacies, research institutes, and universities worldwide.
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Let us handle your sourcing / supply activities. Highly experienced in sourcing specialty raw pharmaceutical ingredients from niche GMP manufacturers around the world.
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Niche API specialist - Pro-active supply partner - High service level - Global network - Logistics according to GDP regulations
Product Description
Mechanism of action
Bisoprolol is a highly selective β₁‑adrenergic receptor antagonist that reduces heart rate, cardiac output and renin release, leading to decreased myocardial oxygen demand and improved haemodynamics. Its β₁ selectivity minimises bronchoconstriction and metabolic interference compared with non-selective β‑blockers.
Benefits and advantages
Widely used in cardiovascular research, heart‑failure modelling, adrenergic‑receptor signalling studies, RAAS regulation experiments, antihypertensive drug-development and electrophysiology of β₁ blockade.
Side effects and risks
Risks include bradycardia, hypotension, fatigue, AV-block progression and rare bronchospasm. Handle with cardiovascular‑active compound precautions.
Datasheet
| Molecular Formula | C40H66N2O12 |
|---|---|
| Molecular Weight | 767.0 g/mol |
| CAS Number | 104344-23-2 |
| Storage Condition | Store at 20 deg to 25 °C (68 deg to 77 °F). Protect from moisture. Dispense in tight containers. |
| Solubility | 7.07e-02 g/L |
| Purity | Purity information is available upon request (COA). |
| Synonym | Bisoprolol fumarate; 104344-23-2; Bisoprolol hemifumarate; Zebeta; Detensiel |
| IUPAC/Chemical Name | (E)-but-2-enedioic acid;bis(1-(propan-2-ylamino)-3-[4-(2-propan-2-yloxyethoxymethyl)phenoxy]propan-2-ol) |
| InChl Key | VMDFASMUILANOL-WXXKFALUSA-N |
| InChl Code | InChI=1S/2C18H31NO4.C4H4O4/c2*1-14(2)19-11-17(20)13-23-18-7-5-16(6-8-18)12-21-9-10-22-15(3)4;5-3(6)1-2-4(7)8/h2*5-8,14-15,17,19-20H,9-13H2,1-4H3;1-2H,(H,5,6)(H,7,8)/b;;2-1+ |
| References |
3D Conformer.
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