AZACYCLONOL
Azapropazone is an NSAID inhibiting prostaglandin synthesis for pain and inflammation management. Benefits include strong anti-inflammatory action. Side effects include gastric irritation, edema, and rare hypersensitivity reactions. Only GMP materials will be supplied, logistics all according to GDP.
About MedicaPharma
MedicaPharma distributes high-quality active pharmaceutical ingredients (APIs) to hospitals, commercial (compounding) pharmacies, research institutes, and universities worldwide.
Network of over +400 GMP API producers
Let us handle your sourcing / supply activities. Highly experienced in sourcing specialty raw pharmaceutical ingredients from niche GMP manufacturers around the world.
Why Choose MedicaPharma
Niche API specialist - Pro-active supply partner - High service level - Global network - Logistics according to GDP regulations
Product Description
Mechanism of action
Azacyclonol is a diphenylmethanol derivative acting mainly as a central antidyskinetic and antipsychotic adjunct. Its mechanism involves antagonism at serotonin 5HT2 receptors and partial antihistaminic and anticholinergic activity. Historically, it was used to reduce hallucinations caused by LSD and other serotonergic hallucinogens.
Benefits and advantages
Important in neuropharmacology for studying serotonergic modulation, psychotomimetic reversal, sensory integration, and antihistaminic/anticholinergic interactions. Also used as a tool compound for mapping cortical serotonin pathways.
Side effects and risks
Potential sedation, dizziness, anticholinergic burden, QT prolongation and CNS depression. Handle with neuroactivecompound PPE.
Only GMP materials will be supplied, logistics all according to GDP.
Datasheet
| Molecular Formula | C17H23NO |
|---|---|
| Molecular Weight | 267.4 g/mol |
| CAS Number | 115-46-8 |
| Storage Condition | Store in a cool, dry place. Keep container tightly closed. Protect from moisture and light. |
| Solubility | >40.1 [ug/mL] (The mean of the results at pH 7.4) |
| Purity | Purity information is available upon request (COA). |
| Synonym | Azacyclonol; 115-46-8; diphenyl(piperidin-4-yl)methanol; gamma-Pipradol; Azaciclonolo |
| IUPAC/Chemical Name | diphenyl(piperidin-4-yl)methanol |
| InChl Key | ZMISODWVFHHWNR-UHFFFAOYSA-N |
| InChl Code | InChI=1S/C18H21NO/c20-18(15-7-3-1-4-8-15,16-9-5-2-6-10-16)17-11-13-19-14-12-17/h1-10,17,19-20H,11-14H2 |
| References |
3D Conformer.
(Click, turn or enlarge)
Download our GMP API Product List.
MedicaPharma is an EU-based supplier of GMP-certified APIs that serves leading healthcare institutions and research organizations.
Click here to download our full API product list.
