About MedicaPharma
MedicaPharma distributes high-quality active pharmaceutical ingredients (APIs) to hospitals, commercial (compounding) pharmacies, research institutes, and universities worldwide.
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Let us handle your sourcing / supply activities. Highly experienced in sourcing specialty raw pharmaceutical ingredients from niche GMP manufacturers around the world.
Why Choose MedicaPharma
Niche API specialist - Pro-active supply partner - High service level - Global network - Logistics according to GDP regulations
Product Description
Mechanism of action
Aminopropylone is an amino‑ketone derivative functioning as a voltage-gated sodium channel blocker. By binding to the intracellular portion of the Naᵥ channel, it stabilises the inactivated state and suppresses initiation and conduction of neuronal action potentials.
Benefits and advantages
Valuable in electrophysiology, anaesthetic analogue research and comparative nerve-block studies. Its unique structure contributes to SAR datasets for synthetic anaesthetic development.
Side effects and risks
Potential cardiotoxicity, CNS excitation, seizure induction and respiratory depression at high concentrations. Stringent anaesthetic-grade handling procedures required.
Datasheet
| Molecular Formula | C16H22N4O2 |
|---|---|
| Molecular Weight | 302.37 g/mol |
| CAS Number | 653884 |
| Storage Condition | Store in a cool, dry place. Keep container tightly closed. Protect from moisture and light. |
| Solubility | Solubility depends on solvent and conditions (e.g., pH). Please contact us for solvent-specific guidance. |
| Purity | Purity information is available upon request (COA). |
| Synonym | Aminopropylon; amipylo; 3690-04-8; aminopropyron; JB5F72V65T |
| IUPAC/Chemical Name | 2-(dimethylamino)-N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)propanamide |
| InChl Key | UQNCVOXEVRELFR-UHFFFAOYSA-N |
| InChl Code | InChI=1S/C16H22N4O2/c1-11-14(17-15(21)12(2)18(3)4)16(22)20(19(11)5)13-9-7-6-8-10-13/h6-10,12H,1-5H3,(H,17,21) |
| References |
3D Conformer.
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