CYPROTERONE ACETATE
Cyproheptadine HCl is an antihistamine blocking H1 receptors, also used to stimulate appetite. Side effects include drowsiness, dry mouth, and weight gain.
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Product Description
Mechanism of Action
Cyproterone acetate is a steroidal antiandrogen that competes with dihydrotestosterone (DHT) at androgen receptors and suppresses gonadotropin release via progesterone‑like negative feedback. It reduces androgen‑dependent growth and signalling.
Benefits and Advantages
Used in androgen‑receptor studies, hormone‑suppression modelling, endocrine‑disorder research, and antiandrogenic compound SAR analysis.
Side Effects and Risks
Risks include hepatotoxicity, thromboembolic events, fatigue, gynecomastia, mood changes and endocrine disturbance. Handle with hormone‑modulating‑agent precautions.
Datasheet
| Molecular Formula | C24H29ClO4 |
|---|---|
| Molecular Weight | 416.9 g/mol |
| CAS Number | 427-51-0 |
| Storage Condition | Keep container tightly closed in a dry and well-ventilated place. Recommended storage temperature: 2 – 8 °C |
| Solubility | Very soluble in dichloromethane and acetone; soluble in methanol; sparingly soluble in ethanol. |
| Purity | Purity information is available upon request (COA). |
| Synonym | CYPROTERONE ACETATE; 427-51-0; Androcur; Cyproterone 17-O-acetate; Cyprostat |
| IUPAC/Chemical Name | [(1S,2S,3S,5R,11R,12S,15R,16S)-15-acetyl-9-chloro-2,16-dimethyl-6-oxo-15-pentacyclo[9.7.0.02,8.03,5.012,16]octadeca-7,9-dienyl] acetate |
| InChl Key | UWFYSQMTEOIJJG-FDTZYFLXSA-N |
| InChl Code | InChI=1S/C24H29ClO4/c1-12(26)24(29-13(2)27)8-6-16-14-10-20(25)19-11-21(28)15-9-18(15)23(19,4)17(14)5-7-22(16,24)3/h10-11,14-18H,5-9H2,1-4H3/t14-,15+,16-,17-,18-,22-,23-,24-/m0/s1 |
| References |
3D Conformer.
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