CARAMIPHEN EDISYLATE

Caramiphen edisylate is an anticholinergic and antitussive used to suppress cough and reduce secretions. Side effects include dry mouth, dizziness, and drowsiness. Only GMP materials will be supplied, logistics all according to GDP.

SKU: b0db310f78fa Category: Tag:

Product Description


Mechanism of action

Caramiphen is a centrally acting antitussive and anticholinergic agent. It suppresses medullary coughcentre excitability while blocking muscarinic receptors in the CNS and peripheral tissues. It also exhibits weak antihistaminic activity and reduces upper airway secretions.

Benefits and advantages

Used in coughreflex physiology studies, vagalafferent inhibition modelling, muscarinicreceptor pharmacology, antitussive SAR investigations and CNSrespiratory control research.

Side effects and risks

Risks include anticholinergic effects (dry mouth, blurred vision, urinary retention), dizziness, tachycardia and mild sedation. Handle with CNSactive antimuscarinic precautions.

Only GMP materials will be supplied, logistics all according to GDP.

Datasheet


Molecular Formula

C38H60N2O10S2

Molecular Weight

769.0 g/mol

CAS Number

22316-47-8

Storage Condition

Store tablets and oral suspension at 20 °C to 25 °C (68 °F to 77 °F).

Solubility

Solubility depends on solvent and conditions (e.g., pH). Please contact us for solvent-specific guidance.

Purity

Purity information is available upon request (COA).

Synonym

Caramiphen edisylate; Caramiphen ethanedisulfonate; 125-86-0; 09TQU5PG95; DTXSID9047835

IUPAC/Chemical Name

bis(2-(diethylamino)ethyl 1-phenylcyclopentane-1-carboxylate);ethane-1,2-disulfonic acid

InChl Key

BANIDACEBXZGNK-UHFFFAOYSA-N

InChl Code

InChI=1S/2C18H27NO2.C2H6O6S2/c2*1-3-19(4-2)14-15-21-17(20)18(12-8-9-13-18)16-10-6-5-7-11-16;3-9(4,5)1-2-10(6,7)8/h2*5-7,10-11H,3-4,8-9,12-15H2,1-2H3;1-2H2,(H,3,4,5)(H,6,7,8)

References

https://pubchem.ncbi.nlm.nih.gov/compound/517304;

3D Conformer.

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