RAXOATIDINE ACETATE

Raxotidine acetate provides improved stability with similar H2blocking effects. Side effects include fatigue, constipation, dizziness, and rare hypersensitivity. Only GMP materials will be supplied, logistics all according to GDP.

SKU: 25931eb16d84 Category: Tag:

Product Description


Mechanism of Action

RAXOATIDINE ACETATE displays a multidimensional biochemical activity profile integrating modulation of enzymatic pathways, receptormediated signalling, mitochondrial bioenergetics, oxidativestress homeostasis, ionchannel dynamics, membrane structural behaviour and transcriptionfactor regulation. Structural modelling suggests interactions with catalytic residues, allosteric microdomains, transmembrane helices, signalling cofactors and cytoskeletal complexes. These interactions enable influence over phosphorylation cascades, secondmessenger flux (Ca²⁺, IP, DAG, cAMP), ROS balance, ATP turnover, membranepotential stability and organelle stressresponse thresholds.

Benefits and Applications

  • Receptorligand affinity analysis and docking studies
  • Enzymekinetic profiling and catalyticflux pathway mapping
  • Mitochondrialfunction modelling and ATP/ROS system evaluation
  • Transcriptomic, metabolomic, proteomic and phosphoproteomic profiling
  • Cytoskeletalarchitecture and membranedynamics exploration
  • Apoptosis, autophagy, necroptosis and ferroptosis pathway modelling
  • SAR/QSAR modelling and compoundoptimisation workflows
  • Mechanistic pharmacodynamics and doseresponse simulation

Side Effects and Risks

  • Oxidativestress imbalance and elevated ROS
  • Mitochondrial overload or respiratorychain suppression
  • Disruption of Ca²⁺/Na⁺/K⁺ ionhomeostasis
  • Unintended receptor crosstalk or inhibitory signal interference
  • Cytoskeletal destabilisation and membrane-integrity reduction
  • Dosedependent cytotoxicity or programmed-cell-death activation
  • Transcriptional and epigenetic instability
  • Inflammatorycascade activation (NF-κB, MAPK, JNK)

Only GMP materials will be supplied, logistics all according to GDP.

Datasheet


Molecular Weight

g/mol

Storage Condition

Store at 2-8°C

Solubility

Soluble in water

Purity

Purity information is available upon request (COA).

IUPAC/Chemical Name

Raxotidine acetate

InChl Key

Unavailable

InChl Code

Unavailable

References

PubChem; ChemBL; FDA;

3D Conformer.

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