MEPHENESIN

Mephenesin is a centrally acting muscle relaxant reducing nerve transmission. Benefits include relief of muscle spasms. Side effects include drowsiness, hypotension, and respiratory depression. Only GMP materials will be supplied, logistics all according to GDP.

SKU: e7d3a5dccb31 Category: Tag:

Product Description


Mechanism of Action

MEPHENESIN displays a broad and multiaxis biochemical interaction profile characterised by modulation of enzymatic networks, receptormediated signalling, intracellular ion regulation, mitochondrial bioenergetics and transcriptional pathway governance. Its structural features suggest interactions with catalytic and regulatory proteins, leading to changes in phosphorylation cycles, metabolic flux, mitochondrial redox balance, calciumsignalling behaviour and stressresponse activation. Depending on cellular environment and concentration, the compound may act as an activator, inhibitor or regulatory modulator.

Benefits and Advantages

This compound supports a wide range of , including:

  • Receptorligand affinity profiling and bindingsite mapping
  • Enzymecascade modelling and catalyticdomain interaction studies
  • Mitochondrialfunction assays, oxidativestress evaluation and metabolicflux tracking
  • Transcriptomic, proteomic and metabolomic investigation for pathway mapping
  • Apoptosis / autophagy pathway research and cellularstress modelling
  • Highresolution mechanismofaction studies and SAR exploration

Side Effects and Risks

Potential risks include oxidative imbalance, mitochondrial overload, ionchannel dysregulation, receptor crosstalk, cytoskeletal disruption and dosedependent cytotoxicity. At elevated exposure levels, the compound may induce apoptosis, autophagy, inflammatory signalling, metabolic reprogramming or transcriptional instability. Proper laboratory controls and strict biosafety procedures are required for handling.

Only GMP materials will be supplied, logistics all according to GDP.

Datasheet


Molecular Formula

C10H14O3

Molecular Weight

182.22 g/mol

CAS Number

59-47-2

Storage Condition

Store in a cool, dry place. Keep container tightly closed. Protect from moisture and light.

Solubility

Sparingly soluble

Purity

Purity information is available upon request (COA).

Synonym

mephenesin; 59-47-2; Mephenesine; Tolserol; Cresoxydiol

IUPAC/Chemical Name

3-(2-methylphenoxy)propane-1,2-diol

InChl Key

JWDYCNIAQWPBHD-UHFFFAOYSA-N

InChl Code

InChI=1S/C10H14O3/c1-8-4-2-3-5-10(8)13-7-9(12)6-11/h2-5,9,11-12H,6-7H2,1H3

References

https://pubchem.ncbi.nlm.nih.gov/compound/4059;

3D Conformer.

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