MEPENZOLATE BROMIDE

Mepenzolate bromide is an anticholinergic reducing GI spasms and secretions. Benefits include relief in peptic ulcer and IBS. Side effects include dry mouth, blurred vision, constipation, and urinary retention.

SKU: 75dd5a2f7ff3 Category: Tag:

Product Description


Mechanism of Action

MEPENZOLATE BROMIDE (ID 26642) displays a broad and multi‑axis biochemical interaction profile characterised by modulation of enzymatic networks, receptor‑mediated signalling, intracellular ion regulation, mitochondrial bioenergetics and transcriptional pathway governance. Its structural features suggest interactions with catalytic and regulatory proteins, leading to changes in phosphorylation cycles, metabolic flux, mitochondrial redox balance, calcium‑signalling behaviour and stress‑response activation. Depending on cellular environment and concentration, the compound may act as an activator, inhibitor or regulatory modulator.

Benefits and Advantages

This compound supports a wide range of research applications, including:

  • Receptor–ligand affinity profiling and binding‑site mapping
  • Enzyme‑cascade modelling and catalytic‑domain interaction studies
  • Mitochondrial‑function assays, oxidative‑stress evaluation and metabolic‑flux tracking
  • Transcriptomic, proteomic and metabolomic investigation for pathway mapping
  • Apoptosis / autophagy pathway research and cellular‑stress modelling
  • High‑resolution mechanism‑of‑action studies and SAR exploration

Side Effects and Risks

Potential risks include oxidative imbalance, mitochondrial overload, ion‑channel dysregulation, receptor cross‑talk, cytoskeletal disruption and dose‑dependent cytotoxicity. At elevated exposure levels, the compound may induce apoptosis, autophagy, inflammatory signalling, metabolic reprogramming or transcriptional instability. Proper laboratory controls and strict biosafety procedures are required for handling.

Datasheet


Molecular Formula

C21H26BrNO3

Molecular Weight

420.3 g/mol

CAS Number

76-90-4

Storage Condition

Store in a cool, dry place. Keep container tightly closed. Protect from moisture and light.

Solubility

>63.1 [ug/mL] (The mean of the results at pH 7.4)

Purity

Purity information is available upon request (COA).

Synonym

MEPENZOLATE BROMIDE; 76-90-4; Cantil; Bromure de mepenzolate; Bromuro de mepenzolato

IUPAC/Chemical Name

(1,1-dimethylpiperidin-1-ium-3-yl) 2-hydroxy-2,2-diphenylacetate bromide

InChl Key

JRRNZNSGDSFFIR-UHFFFAOYSA-M

InChl Code

InChI=1S/C21H26NO3.BrH/c1-22(2)15-9-14-19(16-22)25-20(23)21(24,17-10-5-3-6-11-17)18-12-7-4-8-13-18;/h3-8,10-13,19,24H,9,14-16H2,1-2H3;1H/q+1;/p-1

References

https://pubchem.ncbi.nlm.nih.gov/compound/6461;

3D Conformer.

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