IMIPRAMINE PAMOATE

Imipramine pamoate is a longacting tricyclic antidepressant that enhances serotonin and norepinephrine levels to treat depression and anxiety. Side effects include dry mouth, dizziness, constipation, and potential cardiac rhythm disturbances. Only GMP materials will be supplied, logistics all according to GDP.

SKU: b365394b21be Category: Tag:

Product Description


Mechanism of Action

IMIPRAMINE PAMOATE exhibits a multi-dimensional biochemical activity profile that affects cellular regulation at enzyme, receptor, and transcriptional levels. Its molecular interactions can alter phosphorylation cycles, modulate ionic homeostasis, influence mitochondrial respiration, and adjust redox-signaling pathways. Structural properties suggest specific affinity for regulatory proteins, enabling modulation of metabolic flux and cellular response thresholds.

Benefits and Advantages

This compound is suited for high-resolution mechanistic research, multiomics integration studies, receptor-binding experiments, enzyme-pathway mapping, and advanced pharmacodynamic modelling. It supports ROS-regulation assays, signalling-cascade analysis, cytoskeletaldynamics research, and metabolic adaptation models. Due to predictable biochemical behaviour, it is often used as a comparative reference in pathwayperturbation studies.

  • Useful in mechanistic pharmacology and biochemical modelling
  • Applicable in oxidative-stress, mitochondrial-function and signalling studies
  • Reliable for transcriptional and proteomic profiling
  • Supports SAR (structureactivity relationship) investigations

Side Effects and Risks

Potential risks include mitochondrial overload, ROS imbalance, inadvertent receptor crosstalk, disruption of ion-channel dynamics, and dose-dependent cytotoxicity. High exposure may trigger apoptosis, autophagy, or cellular stress-response activation. Controlled handling conditions and biosafety protocols are required for laboratory use.

Only GMP materials will be supplied, logistics all according to GDP.

Datasheet


Molecular Formula

C19H24N2·C23H16O6

Molecular Weight

949.2 g/mol

CAS Number

10075-24-8

Storage Condition

Store in a cool, dry place. Keep container tightly closed. Protect from moisture and light.

Solubility

Solubility depends on solvent and conditions (e.g., pH). Please contact us for solvent-specific guidance.

Purity

Purity information is available upon request (COA).

Synonym

Imipramine pamoate; 10075-24-8; Tofranil-PM; Imipramine embonate; MC34P30298

IUPAC/Chemical Name

4-[(3-carboxy-2-hydroxynaphthalen-1-yl)methyl]-3-hydroxynaphthalene-2-carboxylic acid;bis(3-(5,6-dihydrobenzo[b][1]benzazepin-11-yl)-N,N-dimethylpropan-1-amine)

InChl Key

BPQZYOJIXDMZSX-UHFFFAOYSA-N

InChl Code

InChI=1S/C23H16O6.2C19H24N2/c24-20-16(14-7-3-1-5-12(14)9-18(20)22(26)27)11-17-15-8-4-2-6-13(15)10-19(21(17)25)23(28)29;2*1-20(2)14-7-15-21-18-10-5-3-8-16(18)12-13-17-9-4-6-11-19(17)21/h1-10,24-25H,11H2,(H,26,27)(H,28,29);2*3-6,8-11H,7,12-15H2,1-2H3

References

https://pubchem.ncbi.nlm.nih.gov/compound/24904;

3D Conformer.

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