IMIPRAMINE PAMOATE

Imipramine pamoate is a long‑acting tricyclic antidepressant that enhances serotonin and norepinephrine levels to treat depression and anxiety. Side effects include dry mouth, dizziness, constipation, and potential cardiac rhythm disturbances.

SKU: b365394b21be Category: Tag:

Product Description


Mechanism of Action

IMIPRAMINE PAMOATE (ID 26414) exhibits a multi-dimensional biochemical activity profile that affects cellular regulation at enzyme, receptor, and transcriptional levels. Its molecular interactions can alter phosphorylation cycles, modulate ionic homeostasis, influence mitochondrial respiration, and adjust redox-signaling pathways. Structural properties suggest specific affinity for regulatory proteins, enabling modulation of metabolic flux and cellular response thresholds.

Benefits and Advantages

This compound is suited for high-resolution mechanistic research, multi‑omics integration studies, receptor-binding experiments, enzyme-pathway mapping, and advanced pharmacodynamic modelling. It supports ROS-regulation assays, signalling-cascade analysis, cytoskeletal‑dynamics research, and metabolic adaptation models. Due to predictable biochemical behaviour, it is often used as a comparative reference in pathway‑perturbation studies.

  • Useful in mechanistic pharmacology and biochemical modelling
  • Applicable in oxidative-stress, mitochondrial-function and signalling studies
  • Reliable for transcriptional and proteomic profiling
  • Supports SAR (structure–activity relationship) investigations

Side Effects and Risks

Potential risks include mitochondrial overload, ROS imbalance, inadvertent receptor cross‑talk, disruption of ion-channel dynamics, and dose-dependent cytotoxicity. High exposure may trigger apoptosis, autophagy, or cellular stress-response activation. Controlled handling conditions and biosafety protocols are required for laboratory use.

Datasheet


Molecular Formula

C19H24N2·C23H16O6

Molecular Weight

949.2 g/mol

CAS Number

10075-24-8

Storage Condition

Store in a cool, dry place. Keep container tightly closed. Protect from moisture and light.

Solubility

Solubility depends on solvent and conditions (e.g., pH). Please contact us for solvent-specific guidance.

Purity

Purity information is available upon request (COA).

Synonym

Imipramine pamoate; 10075-24-8; Tofranil-PM; Imipramine embonate; MC34P30298

IUPAC/Chemical Name

4-[(3-carboxy-2-hydroxynaphthalen-1-yl)methyl]-3-hydroxynaphthalene-2-carboxylic acid;bis(3-(5,6-dihydrobenzo[b][1]benzazepin-11-yl)-N,N-dimethylpropan-1-amine)

InChl Key

BPQZYOJIXDMZSX-UHFFFAOYSA-N

InChl Code

InChI=1S/C23H16O6.2C19H24N2/c24-20-16(14-7-3-1-5-12(14)9-18(20)22(26)27)11-17-15-8-4-2-6-13(15)10-19(21(17)25)23(28)29;2*1-20(2)14-7-15-21-18-10-5-3-8-16(18)12-13-17-9-4-6-11-19(17)21/h1-10,24-25H,11H2,(H,26,27)(H,28,29);2*3-6,8-11H,7,12-15H2,1-2H3

References

https://pubchem.ncbi.nlm.nih.gov/compound/24904;

3D Conformer.

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