GESTRINONE

Gestrinone is a steroidal agent with antiestrogenic and antiprogestogenic effects used in endometriosis. Side effects include acne, weight gain, and voice changes. Only GMP materials will be supplied, logistics all according to GDP.

SKU: d3be030a01a3 Category: Tag:

Product Description


Mechanism of Action

Gestrinone is a synthetic steroid with mixed progestogenic, antiestrogenic and androgenic activity, modulating multiple hormone receptors and suppressing endometrial proliferation.

Benefits and Advantages

Used in endocrine-pathway modelling, receptor-binding assays, reproductive research and estrogen-antagonism studies.

Side Effects and Risks

Acne, weight changes, masculinization effects and hormonal fluctuations.

Only GMP materials will be supplied, logistics all according to GDP.

Datasheet


Molecular Formula

C21H24O2

Molecular Weight

308.4 g/mol

CAS Number

16320-04-0

Storage Condition

Store in a cool, dry place. Keep container tightly closed. Protect from moisture and light.

Solubility

Solubility depends on solvent and conditions (e.g., pH). Please contact us for solvent-specific guidance.

Purity

Purity information is available upon request (COA).

Synonym

Gestrinone; 16320-04-0; Dimetriose; Ethylnorgestrienone; Gestrinona

IUPAC/Chemical Name

(8S,13S,14S,17R)-13-ethyl-17-ethynyl-17-hydroxy-1,2,6,7,8,14,15,16-octahydrocyclopenta[a]phenanthren-3-one

InChl Key

BJJXHLWLUDYTGC-ANULTFPQSA-N

InChl Code

InChI=1S/C21H24O2/c1-3-20-11-9-17-16-8-6-15(22)13-14(16)5-7-18(17)19(20)10-12-21(20,23)4-2/h2,9,11,13,18-19,23H,3,5-8,10,12H2,1H3/t18-,19+,20+,21+/m1/s1

References

https://pubchem.ncbi.nlm.nih.gov/compound/27812;

3D Conformer.

(Click, turn or enlarge)

Download our GMP API Product List.

MedicaPharma is an EU-based supplier of GMP-certified APIs that serves leading healthcare institutions and research organizations.
Click here to download our full API product list.

Download