About MedicaPharma
MedicaPharma distributes high-quality active pharmaceutical ingredients (APIs) to hospitals, commercial (compounding) pharmacies, research institutes, and universities worldwide.
Network of over +400 GMP API producers
Let us handle your sourcing / supply activities. Highly experienced in sourcing specialty raw pharmaceutical ingredients from niche GMP manufacturers around the world.
Why Choose MedicaPharma
Niche API specialist - Pro-active supply partner - High service level - Global network - Logistics according to GDP regulations
Product Description
Mechanism of Action
Epinastine hydrochloride is a dual Hhistamine receptor antagonist and mastcell stabilizer. It prevents histamine release and blocks downstream allergicinflammation pathways without significant CNS penetration.
Benefits and Advantages
Used in allergicinflammation modelling, Hreceptor antagonism assays, mastcell mediator studies, and ocularantiallergy pharmacology.
Side Effects and Risks
Risks include headache, ocular irritation (topical forms), dry eyes, and rare hypersensitivity reactions. Handle with antihistamineclass precautions.
Only GMP materials will be supplied, logistics all according to GDP.
Datasheet
| Molecular Formula | C16H16N4·HCl |
|---|---|
| Molecular Weight | 285.77 g/mol |
| CAS Number | 108929-04-0 |
| Storage Condition | Store in a cool, dry place. Keep container tightly closed. Protect from moisture and light. |
| Solubility | Solubility depends on solvent and conditions (e.g., pH). Please contact us for solvent-specific guidance. |
| Purity | Purity information is available upon request (COA). |
| Synonym | Epinastine hydrochloride; 108929-04-0; Epinastine HCl; Alesion; Elestat |
| IUPAC/Chemical Name | 2,4-diazatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),3,7,9,11,14,16-heptaen-3-amine;hydrochloride |
| InChl Key | VKXSGUIOOQPGAF-UHFFFAOYSA-N |
| InChl Code | InChI=1S/C16H15N3.ClH/c17-16-18-10-15-13-7-3-1-5-11(13)9-12-6-2-4-8-14(12)19(15)16;/h1-8,15H,9-10H2,(H2,17,18);1H |
| References |
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