CARTEOLOL

Carteolol is a nonselective betablocker used in ophthalmology to lower intraocular pressure in glaucoma. Side effects include eye irritation, blurred vision, and rare bradycardia. Only GMP materials will be supplied, logistics all according to GDP.

SKU: 8f9893de3992 Category: Tag:

Product Description


Mechanism of action

Carteolol is a nonselective adrenergic receptor antagonist with intrinsic sympathomimetic activity. It reduces intraocular pressure by decreasing aqueoushumor production and enhancing outflow. In systemic tissues it decreases heart rate, contractility and renin secretion.

Benefits and advantages

Used in glaucoma research, receptor pharmacology, aqueoushumor dynamics studies, cardiovascular blocker modelling and sympathomimeticactivity investigations.

Side effects and risks

Risks include bradycardia, bronchoconstriction, hypotension, fatigue and ocular irritation. Handle with betablocker safety precautions.

Only GMP materials will be supplied, logistics all according to GDP.

Datasheet


Molecular Formula

C16H24N2O3

Molecular Weight

292.37 g/mol

CAS Number

51781-06-7

Storage Condition

Store in a cool, dry place. Keep container tightly closed. Protect from moisture and light.

Solubility

4.21e-01 g/L

Purity

Purity information is available upon request (COA).

Synonym

CARTEOLOL; 51781-06-7; Carteololum; 8NF31401XG; 2(1H)-Quinolinone, 5-(3-((1,1-dimethylethyl)amino)-2-hydroxypropoxy)-3,4-dihydro-

IUPAC/Chemical Name

5-[3-(tert-butylamino)-2-hydroxypropoxy]-3,4-dihydro-1H-quinolin-2-one

InChl Key

LWAFSWPYPHEXKX-UHFFFAOYSA-N

InChl Code

InChI=1S/C16H24N2O3/c1-16(2,3)17-9-11(19)10-21-14-6-4-5-13-12(14)7-8-15(20)18-13/h4-6,11,17,19H,7-10H2,1-3H3,(H,18,20)

References

https://pubchem.ncbi.nlm.nih.gov/compound/2583;

3D Conformer.

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