CIMETROPIUM BROMIDE

Cimetropium bromide is an anticholinergic reducing GI motility and secretions, used for IBS and abdominal cramps. Side effects include dry mouth, blurred vision, and constipation. Only GMP materials will be supplied, logistics all according to GDP.

SKU: a0882535ca25 Category: Tag:

Product Description


Mechanism of Action

Cimetropium bromide is a quaternary ammonium antimuscarinic agent that blocks M muscarinic receptors on smooth muscle. This reduces gastric motility, intestinal spasms and secretions. Due to poor bloodbrain barrier penetration, it primarily acts peripherally without strong CNS effects.

Benefits and Advantages

Used in GIspasm research, muscarinicreceptor pharmacology, smoothmuscle contractility studies, anticholinergic SAR investigations and functional boweldisorder modelling.

Side Effects and Risks

Risks include dry mouth, constipation, blurred vision, urinary retention and tachycardia. Handle using antimuscarinicagent precautions.

Only GMP materials will be supplied, logistics all according to GDP.

Datasheet


Molecular Formula

C21H38BrNO5

Molecular Weight

438.4 g/mol

CAS Number

51598-60-8

Storage Condition

Store in a cool, dry place. Keep container tightly closed. Protect from moisture and light.

Solubility

Solubility depends on solvent and conditions (e.g., pH). Please contact us for solvent-specific guidance.

Purity

Purity information is available upon request (COA).

Synonym

Cimetropium Bromide; Cimetropium (Bromide); Bromuro de cimetropio; Alginor; Bromure de cimetropium

IUPAC/Chemical Name

[(1R,2R,4S,5S)-9-(cyclopropylmethyl)-9-methyl-3-oxa-9-azoniatricyclo[3.3.1.02,4]nonan-7-yl] (2S)-3-hydroxy-2-phenylpropanoate bromide

InChl Key

WDURTRGFUGAJHA-HNHWXVNLSA-M

InChl Code

InChI=1S/C21H28NO4.BrH/c1-22(11-13-7-8-13)17-9-15(10-18(22)20-19(17)26-20)25-21(24)16(12-23)14-5-3-2-4-6-14;/h2-6,13,15-20,23H,7-12H2,1H3;1H/q+1;/p-1/t15?,16-,17-,18+,19-,20+,22?;/m1./s1

References

PubChem; ChemBL; FDA;

3D Conformer.

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