ALARELIN

Alarelin is a synthetic GnRH agonist that initially stimulates and later suppresses gonadotropin release. It is used in reproductive research and hormoneregulated conditions. Benefits include precise hormonal modulation. Side effects may include hot flashes, mood changes, and decreased libido. Only GMP materials will be supplied, logistics all according to GDP.

SKU: fa77bdd59978 Category: Tag:

Product Description


Mechanism of action

ALARELIN is a pharmacologically active compound used in specialised medical or biochemical applications. Its mechanism of action involves modulation of specific cellular pathways, receptor interactions or enzyme systems depending on its structural class. In professional environments it is applied to influence defined metabolic, neurological, endocrine or immunological processes.

Benefits and advantages

ALARELIN is valued for its predictable biochemical behaviour, defined purity profile and suitability for advanced formulation or research use. It provides targeted activity relevant to its therapeutic or analytical category, offering consistent performance under controlled conditions. The compound is often incorporated into protocols requiring high specificity or reproducibility.

Side effects and risks

Potential risks depend on the pharmacological class of ALARELIN. These may include organspecific toxicity, allergic reactions, metabolic disturbances or interactions with other active substances. Because potency and toxicity can vary, handling and use are strictly limited to trained professionals operating within regulated laboratory or manufacturing settings.

Only GMP materials will be supplied, logistics all according to GDP.

Datasheet


Molecular Formula

C56H78N16O12

Molecular Weight

1167.3 g/mol

CAS Number

148029-26-9

Storage Condition

Store in a cool, dry place. Keep container tightly closed. Protect from moisture and light.

Solubility

Solubility depends on solvent and conditions (e.g., pH). Please contact us for solvent-specific guidance.

Purity

Purity information is available upon request (COA).

Synonym

ALARELIN; Dalarelin; NJS328SUA7; TAP-127; L-4513

IUPAC/Chemical Name

(2S)-N-[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2R)-1-[[(2S)-1-[[(2S)-5-(diaminomethylideneamino)-1-[(2S)-2-(ethylcarbamoyl)pyrrolidin-1-yl]-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-1-oxopropan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]amino]-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]-5-oxopyrrolidine-2-carboxamide

InChl Key

QLGKMLRGKPKGKI-QWQCQAQZSA-N

InChl Code

InChI=1S/C56H78N16O12/c1-5-60-54(83)45-13-9-21-72(45)55(84)39(12-8-20-61-56(57)58)66-50(79)40(22-30(2)3)67-47(76)31(4)64-49(78)41(23-32-14-16-35(74)17-15-32)68-53(82)44(28-73)71-51(80)42(24-33-26-62-37-11-7-6-10-36(33)37)69-52(81)43(25-34-27-59-29-63-34)70-48(77)38-18-19-46(75)65-38/h6-7,10-11,14-17,26-27,29-31,38-45,62,73-74H,5,8-9,12-13,18-25,28H2,1-4H3,(H,59,63)(H,60,83)(H,64,78)(H,65,75)(H,66,79)(H,67,76)(H,68,82)(H,69,81)(H,70,77)(H,71,80)(H4,57,58,61)/t31-,38+,39+,40+,41+,42+,43+,44+,45+/m1/s1

References

https://pubchem.ncbi.nlm.nih.gov/compound/9855027;

3D Conformer.

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